Medicinal Chemistry Conference

MIKIW 2019 Schedule

Friday, April 12, 2019

Time Agenda Item Location
3:00 – 6:00 p.m. • Registration open
• Hotel check-in
Springhill Suites » - Minnesota and Illinois
Quality Inn and Suites » - Iowa
Days Inn » - Wisconsin
7:00 p.m. Welcome reception Arterra Event Gallery

Saturday, April 13, 2019

* ISB = KU Integrated Science Building

Time Agenda Item Location
8:00 – 8:40 a.m. Breakfast and poster setup ISB Atrium
8:40 – 9:00 a.m. Opening remarks ISB Auditorium
  Oral presentation session 1
Moderators: Patrick Ross, Bo Han
ISB Auditorium
9:00 – 9:25 a.m. Yuwen Yin
Blake Peterson lab, KU
Phorbol Carbamates as Novel Tools for Controlling Cellular Signal Transduction
 
9:25 – 9:50 a.m. Arturo L. Aguirre
Robert Kerns lab, UI
Investigating Quinazoline-2,4-dione and Fluoroquinolone Scaffolds for Antibiotic Activity and Metabolic Stability
 
9:50 – 10:15 a.m. Stephanie Blaszczyk
Weiping Tang lab, UW-Madison
S-Adamantyl Group Directed Site-Selective Acylation and Its Applications in the Streamlined Assembly of Oligosaccharides
 
10:15 – 10:40 a.m. Kellan T. Passow
Daniel A. Harki lab, UMN
The Discovery of 4CIN: Indoles as a Platform for Novel Nucleoside Fluorophore Development
 
10:40 – 11:00 a.m. Break ISB Atrium
11:00 a.m. – noon Keynote address
"Inhibitors of HIV-1 Maturation"
Nicholas A. Meanwell, Ph.D., FRSC
Dept. of Chemistry and Molecular Technologies, Bristol-Myers Squibb Research and Development
ISB Auditorium
12:00 – 1:30 p.m. Lunch and poster setup ISB Atrium
  Oral presentation session 2
Moderators: Sahishna Phaniraj, Bo Han
ISB Auditorium
1:30 – 1:55 p.m. Jacob P. Sorrentino
Ryan Altman lab, KU
Fluorinated Dextromethorphan Analogs to Prevent the Formation of Psychoactive Metabolites
 
1:55 – 2:20 p.m. Brian P. David
Terry W. Moore lab, UIC
Structure-Activity Relationship and Evaluation of Non-electrophilic NRF2 Activators in a Diabetic Mouse Model
 
2:20 – 2:45 p.m. Muhammad M. Khalifa
Jennifer E. Golden lab, UW-Madison
Convergent Annulative Platform for the Synthesis of Ring-Fused Quinolinones
 
2:45 – 3:45 p.m. Poster session: Odd numbered posters present ISB Atrium
3:45 – 4:45 p.m. Poster session: Even numbered posters present ISB Atrium
4:45 – 5:15 p.m. Faculty meeting ISB 1160
6:00 – 7:00 p.m. Faculty mixer (open bar) Van Go inc.
7:00 p.m. Formal banquet dinner Van Go inc.

Sunday, April 14, 2019

* ISB = KU Integrated Science Building

Time Agenda Item Location
  Check-out of hotel prior to breakfast Springhill Suites » - Minnesota and Illinois
Quality Inn and Suites » - Iowa
Days Inn » - Wisconsin
8:00 – 8:40 a.m. Breakfast ISB Atrium
  Oral presentation session 3
Moderators: Patrick Ross, Bo Han
ISB Auditorium
8:40 - 9:05 a.m. Erick J. Carlson
Gunda I. Georg lab, UMN
The Discovery and Characterization of Steroidal Blockers of CatSper
 
9:05 - 9:30 a.m. Alanna Condren
Laura Sanchez lab, UIC
Biofilm Inhibition Alters Specialized Metabolism and Increases Virulence in Pseudomonas Aeruginosa
 
9:30 - 9:55 a.m. Sanjay Bhattarai
Michael S. Wolfe lab, KU
Substrate transmembrane mimetic inhibitors of gamma-secretase: probes for chemical structural biology
 
9:55 - 10:20 a.m. Pratik Rajesh Chheda
Robert J. Kerns lab, UI
Allosteric Inhibitors of Apicoplast DNA Polymerase: New Antimalarials That Bind a Novel Allosteric Binding Site
 
10:20 - 10:40 a.m. Break ISB Atrium
  Oral presentation session 4
Moderators: Tomas Smith, Bo Han
ISB Auditorium
10:40 - 11:05 a.m. Matthew Worth
Jiaoyan Jiang lab, UW-Madison
Covalent Inhibitors Target O-GlcNAc Transferase in Cells
 
11:05 - 11:30 a.m. Ozgun Kilic
Cartson Rick Wagner lab, UMN
Nanorings with Engineered Fibronectins for Cancer Therapeutics
 
11:30 - 11:55 a.m. Katherine E. Zink
Laura M. Sanchez lab, UIC
A Novel Imaging Mass Spectrometry Method for Identifying Preventative Approaches in High Grade Serous Ovarian Cancer
 
12:00 p.m. • Concluding remarks
• Box lunch served
• Buses depart
ISB Atrium